BDBM10885 (4R)-4-(ethylamino)-2-(3-methoxypropyl)-1,1-dioxo-2H,3H,4H-1,7,2-thieno[3,2-e][1,2]thiazine-6-sulfonamide::(R)-4-(ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno(3,2-E)-1,2-thiazine-6-sulfonamide 1,1-dioxide::AL-4862::Azopt::Brinzolamide (BRZ)::brinzolamide
SMILES CCN[C@H]1CN(CCCOC)S(=O)(=O)c2sc(cc12)S(N)(=O)=O
InChI Key InChIKey=HCRKCZRJWPKOAR-JTQLQIEISA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 20 hits for monomerid = 10885
Affinity DataKi: 36nMAssay Description:Inhibition of human carbonic anhydrase9 preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of human membrane bound carbonic anhydrase 9 preincubated for 15 mins at room temperature followed by 72 hrs at 4 degC by stopped flow CO2...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory constant against human Carbonic anhydrase IXMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory constant against catalytic domain of human carbonic anhydrase IXMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human carbonic anhydrase IX expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human tumor-associated transmembrane carbonic anhydrase IX.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human cloned carbonic anhydrase isozyme IX, by CO2 hydrase assay method.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human carbonic anhydrase IXMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of catalytic domain of human recombinant CA IXMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against membrane bound tumor associated human carbonic anhydrase IXMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of human CA 9 catalytic domainMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of human catalytic domain carbonic anhydrase 9 by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Inhibition of human CA9 catalytic domain by CO2 hydration methodMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Inhibition of human cloned catalytic domain CA9 by CO2 hydration methodMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair